
Therapeutic Area | MeSH |
|---|---|
| neoplasms | D009369 |
| urogenital diseases | D000091642 |
| Drug common name | Linzagolix choline |
| INN | — |
| Description | Linzagolix, sold under the brand name Yselty, is a medication used in the treatment of uterine fibroids. Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) developed by Kissei Pharmaceutical and ObsEva.
|
| Classification | Small molecule |
| Drug class | gonadotropin releasing hormone (GnRH) receptor antagonists (nonpeptide) |
| Image (chem structure or protein) | ![]() |
| Structure (InChI/SMILES or Protein Sequence) | COc1cc(F)c(-n2c(=O)[nH]c3csc(C(=O)[O-])c3c2=O)cc1OCc1c(OC)ccc(F)c1F.C[N+](C)(C)CCO |
| PDB | — |
| CAS-ID | 935283-04-8 |
| RxCUI | — |
| ChEMBL ID | CHEMBL4298171 |
| ChEBI ID | — |
| PubChem CID | 16656889 |
| DrugBank | — |
| UNII ID | — |
